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Total: 10647
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Unknown
Bacterial dihydrofolate reductase inhibitor
Small molecule
Approved
OTHER
ORAL
Chemical and Drug Induced Liver Injury; Cystinuria; Subarachnoid Hemorrhage
Reducing agent
Small molecule
Approved
OTHER
INJECTION
Esophageal and Gastric Varices
Calcium chelating agent
Small molecule
Approved
OTHER
INJECTION
Neoplasms
Diagnostic agent
Protein
Approved
Unknown
Unknown
Gastrointestinal Hemorrhage; Hypotension, Orthostatic; Idiopathic Pulmonary Fibrosis; Infections; Irritable Bowel Syndrome; Migraine Disorders; Obesity; Adenoma, Islet Cell; Carcinoma, Neuroendocrine; Intestinal Obstruction; Meningioma; Neoplasms; Prostatic Neoplasms, Castration-Resistant; Telangiectasia, Hereditary Hemorrhagic; Thymoma; Acromegaly; Carcinoid Tumor; Carcinoma, Hepatocellular; Diarrhea; Malignant Carcinoid Syndrome; Neuroendocrine Tumors; Pancreatic Neoplasms; Polycystic Kidney, Autosomal Dominant
Unknown
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
INJECTION; INTRAVENOUS; ORAL
Adenocarcinoma; Blastic Plasmacytoid Dendritic Cell Neoplasm; Ganglioneuroblastoma; Kidney Neoplasms; Leukemia, Biphenotypic, Acute; Leukemia, Myeloid, Acute; Muscular Diseases; Myasthenia Gravis; Myelodysplastic Syndromes; Neoplasm Metastasis; Obesity; Osteosarcoma; Primary Myelofibrosis; Stiff-Person Syndrome; Vasculitis; Acute Kidney Injury; Anemia, Aplastic; Anemia, Sickle Cell; Burkitt Lymphoma; Carcinoma, Hepatocellular; Central Nervous System Neoplasms; Crohn Disease; Hematologic Neoplasms; Hodgkin Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Lupus Erythematosus, Systemic; Lymphoma, B-Cell; Lymphoma, Follicular; Lymphoma, Mantle-Cell; Lymphoma, Non-Hodgkin; Melanoma; Multiple Myeloma; Multiple Sclerosis; Neoplasms; Neoplasms, Germ Cell and Embryonal; Neuromyelitis Optica; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Renal Insufficiency, Chronic; Retinoblastoma; Sarcoma, Ewing; Testicular Neoplasms; Brain Neoplasms; Breast Neoplasms; Ependymoma; Leukemia; Leukemia, Lymphoid; Lung Neoplasms; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Medulloblastoma; Multiple Sclerosis, Relapsing-Remitting; Neuroblastoma; Sarcoma; Scleroderma, Systemic; Thrombocytopenia
Unknown
Small molecule
Approved
OTHER
INJECTION
Cicatrix; Cardiomyopathy, Dilated; Hypertension
Angiotensin-converting enzyme inhibitor
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Glaucoma
Unknown
Small molecule
Approved
OTHER
ORAL
Abortion, Incomplete; Infections; Clostridium Infections; Muscle Cramp; Non-alcoholic Fatty Liver Disease; Premature Birth; Abortion, Spontaneous; Leiomyoma; Menorrhagia; Myoma; Obesity; Pain; Postpartum Hemorrhage; Pre-Eclampsia; Pregnancy; Spondylitis, Ankylosing; Uterine Diseases; Duodenal Ulcer; Gastroesophageal Reflux; Hemorrhage; Osteoarthritis; Peptic Ulcer; Stomach Ulcer
Prostanoid EP3 receptor agonist
Small molecule
Approved
Unknown
Unknown
Gastritis; Gastroparesis; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Peptic Ulcer
Histamine H2 receptor antagonist
Small molecule
Approved
OTHER
TRANSDERMAL
Amphetamine-Related Disorders; Schizophrenia; Prostatic Neoplasms; Tobacco Use Disorder; Borderline Personality Disorder; Cocaine-Related Disorders; Depressive Disorder; Depressive Disorder, Major; Parkinson Disease
Monoamine oxidase B inhibitor
Small molecule
Approved
Unknown
Unknown
Pain
Kappa opioid receptor antagonist
Unknown
Approved
OTHER
INTRATHECAL
Unknown
Unknown
Small molecule
Approved
OTHER
ORAL
Hypertension
Sulfonylurea receptor 2, Kir6.2 opener
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Ovarian Neoplasms; Polycystic Ovary Syndrome; Prostatic Neoplasms, Castration-Resistant; Carcinoma; Neoplasms; Prostatic Neoplasms
Androgen Receptor antagonist
Small molecule
Approved
GASTROINTESTINAL; OTHER
ORAL
Alzheimer Disease; Anemia; Anemia, Sickle Cell; Arthritis, Rheumatoid; Carcinoma, Medullary; Central Serous Chorioretinopathy; Child Development Disorders, Pervasive; Chronic Pain; Clostridium Infections; Colitis, Ulcerative; Communicable Diseases; Crohn Disease; Dermatitis, Atopic; Diabetes Mellitus; Diabetes Mellitus, Type 2; Erectile Dysfunction; Glaucoma; Hepatitis B, Chronic; Hepatitis C; Hepatitis C, Chronic; HIV Infections; Laryngomalacia; Melanoma; Mitochondrial Diseases; Muscular Atrophy, Spinal; Neoplasms; Pancreatic Neoplasms; Prostatic Neoplasms; Psoriasis; Pulmonary Disease, Chronic Obstructive; Breast Neoplasms; Carcinoma, Squamous Cell; Colorectal Neoplasms; Gastrinoma; Gastritis; Granuloma; Head and Neck Neoplasms; Idiopathic Pulmonary Fibrosis; Lymphoma; Lymphoma, B-Cell, Marginal Zone; Prostatic Neoplasms, Castration-Resistant; Squamous Cell Carcinoma of Head and Neck; Squamous Intraepithelial Lesions; Ulcer; Zollinger-Ellison Syndrome; Barrett Esophagus; Cough; Cysticercosis; Diabetes Mellitus, Type 1; Dyspepsia; Esophagitis, Peptic; Exocrine Pancreatic Insufficiency; Gastrointestinal Hemorrhage; Helicobacter Infections; Hemorrhage; Multiple Sclerosis, Relapsing-Remitting; Osteoarthritis; Pain; Peripheral Nervous System Diseases; Spondylitis, Ankylosing; Stomach Neoplasms; Wounds and Injuries; Duodenal Ulcer; Esophagitis; Gastroesophageal Reflux; Heartburn; Infections; Peptic Ulcer; Stomach Ulcer
Potassium-transporting ATPase inhibitor
Small molecule
Approved
Unknown
Unknown
Anxiety; Dementia; Obsessive-Compulsive Disorder; Premature Ejaculation; Schizophrenia; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Glioblastoma; Gliosarcoma; Leukoencephalopathy, Progressive Multifocal; Pneumonia, Viral; Respiratory Insufficiency; Severe Acute Respiratory Syndrome; Malaria, Falciparum; Schistosomiasis haematobia; Malaria
Unknown
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Osteomyelitis; Colorectal Neoplasms; Bacterial Infections
Unknown
Small molecule
Approved
Unknown
Unknown
Coronary Artery Disease
Unknown
Small molecule
Approved
Unknown
Unknown
Cystic Fibrosis; Hepatitis C; HIV Infections; Migraine Disorders; Metrorrhagia; Osteoporosis; Neural Tube Defects; Acne Vulgaris
Progesterone receptor agonist
Small molecule
Approved
Unknown
Unknown
Bacterial Infections
Unknown
Small molecule
Approved
OTHER
INJECTION; INTRAVENOUS
Inflammation; Ischemia; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Cardiomyopathies; Coronary Disease; Pain; Respiratory Distress Syndrome; ST Elevation Myocardial Infarction; Takotsubo Cardiomyopathy; Angina, Stable; Atrial Fibrillation; Coronary Stenosis; Myocardial Infarction; Myocardial Ischemia; Neoplasms; Tachycardia, Ventricular; Cardiovascular Diseases; Tachycardia, Paroxysmal; Wolff-Parkinson-White Syndrome
Adenosine receptor agonist
Small molecule
Approved
OTHER
INJECTION; INTRAVENOUS; IV (INFUSION)
Adenocarcinoma, Follicular; Adrenal Cortex Neoplasms; Anus Neoplasms; Appendiceal Neoplasms; Carcinoma, Renal Cell; Carcinoma, Verrucous; HIV Infections; Hypopharyngeal Neoplasms; Insulinoma; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Mantle-Cell; Multiple Myeloma; Neoplasms, Cystic, Mucinous, and Serous; Neoplasms, Plasma Cell; Neuroendocrine Tumors; Parathyroid Neoplasms; Pericardial Effusion; Pleural Effusion; Skin Diseases; Somatostatinoma; Vaginal Neoplasms; Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Bile Duct Neoplasms; Bone Neoplasms; Brain Stem Neoplasms; Breast Neoplasms, Male; Burkitt Lymphoma; Carcinoid Tumor; Carcinoma, Endometrioid; Carcinoma, Intraductal, Noninfiltrating; Carcinoma, Islet Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Carcinosarcoma; Cystadenoma, Serous; Gallbladder Neoplasms; Gastrointestinal Stromal Tumors; Gliosarcoma; Hereditary Breast and Ovarian Cancer Syndrome; Leiomyosarcoma; Leukemia; Leukemia, Myeloid, Acute; Lymphoma, B-Cell; Mesothelioma, Malignant; Myelodysplastic Syndromes; Myeloproliferative Disorders; Nasopharyngeal Neoplasms; Neoplasm Metastasis; Neoplasms, Complex and Mixed; Oligodendroglioma; Osteosarcoma; Pancreatic Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Prostatic Neoplasms; Retinal Neoplasms; Salivary Gland Neoplasms; Stomach Neoplasms; Thrombosis; Thymoma; Ureteral Neoplasms; Uveal Melanoma; Vulvar Neoplasms; Wilms Tumor; Adenocarcinoma of Lung; Anemia; Astrocytoma; Biliary Tract Neoplasms; Brain Neoplasms; Breast Neoplasms; Carcinoma; Carcinoma, Hepatocellular; Carcinoma, Large Cell; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Central Nervous System Neoplasms; Cholangiocarcinoma; Choroid Plexus Neoplasms; Colorectal Neoplasms; Endometrial Neoplasms; Ependymoma; Esophageal Neoplasms; Fallopian Tube Neoplasms; Ganglioneuroblastoma; Genital Neoplasms, Female; Gestational Trophoblastic Disease; Glioblastoma; Glioma; Head and Neck Neoplasms; Hepatoblastoma; Hodgkin Disease; Inflammatory Breast Neoplasms; Kidney Neoplasms; Laryngeal Neoplasms; Leukemia-Lymphoma, Adult T-Cell; Liver Neoplasms; Lung Neoplasms; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Medulloblastoma; Melanoma; Mesothelioma; Mouth Neoplasms; Nasopharyngeal Carcinoma; Neoplasms, Germ Cell and Embryonal; Neuroblastoma; Neuroectodermal Tumors, Primitive; Oropharyngeal Neoplasms; Pain; Paraganglioma; Peripheral Nervous System Diseases; Peritoneal Neoplasms; Prostatic Neoplasms, Castration-Resistant; Retinoblastoma; Retroviridae Infections; Sarcoma; Seminoma; Sex Cord-Gonadal Stromal Tumors; Skin Neoplasms; Small Cell Lung Carcinoma; Squamous Cell Carcinoma of Head and Neck; Testicular Neoplasms; Thyroid Neoplasms; Triple Negative Breast Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Uterine Cervical Neoplasms; Uterine Neoplasms; Carcinoma, Ovarian Epithelial; Neoplasms; Ovarian Neoplasms
DNA inhibitor
Protein
Approved
Unknown
Unknown
Adenomyosis; Carcinoma, Lobular; Hodgkin Disease; Metabolic Syndrome; Primary Ovarian Insufficiency; Salivary Gland Neoplasms; Breast Neoplasms; Infertility; Leiomyoma; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Neoplasms
Unknown
Small molecule
Approved
OTHER
ORAL
Anxiety; Bipolar Disorder; Dementia; Depressive Disorder; Developmental Disabilities; Intellectual Disability; Psychotic Disorders; Schizophrenia
Dopamine D2 receptor antagonist
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Glaucoma
Unknown
Small molecule
Approved
Unknown
Unknown
Atrial Fibrillation; Death, Sudden, Cardiac; Heart Failure; Myocardial Infarction; Ventricular Fibrillation; Arrhythmias, Cardiac
Unknown
Protein
Approved
OTHER
UNKNOWN
HIV Infections; Severe Acute Respiratory Syndrome
Interferon alpha/beta receptor agonist
Small molecule
Approved
OTHER
ORAL
Unknown
Beta-1 adrenergic receptor antagonist
Protein
Approved
Unknown
Unknown
Anemia, Sickle Cell; Asphyxia; Diabetic Foot; Substance-Related Disorders; Anemia, Neonatal; beta-Thalassemia; Coronary Disease; Friedreich Ataxia; Myocardial Infarction; Neoplasms; Pancreatic Neoplasms; Peripheral Nervous System Diseases; Premature Birth; ST Elevation Myocardial Infarction; Stroke; Brain Injuries; Breast Neoplasms; Carcinoma, Squamous Cell; Fatigue; Head and Neck Neoplasms; Heart Arrest; Hepatitis C; Hypoxia-Ischemia, Brain; Leukemia; Leukemia, Myeloid, Acute; Lung Neoplasms; Ovarian Neoplasms; Peritoneal Neoplasms; Prostatic Neoplasms; Uterine Cervical Neoplasms; Venous Thrombosis; Anemia; Blood Transfusion, Autologous; HIV Infections; Kidney Failure, Chronic; Myelodysplastic Syndromes; Renal Insufficiency, Chronic
Erythropoietin receptor agonist
Small molecule
Approved
OTHER
ORAL
Neoplasms; Osteomyelitis; HIV Infections; Liver Abscess; Syphilis; Bacterial Infections; Bronchitis; Bronchitis, Chronic; Gonorrhea; Infections; Otitis Media; Pharyngitis; Tonsillitis; Urinary Tract Infections
Bacterial penicillin-binding protein inhibitor