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Total: 10647
Protein
Approved
Unknown
Unknown
Arthritis, Rheumatoid; Renal Insufficiency, Chronic; Diabetes Mellitus, Type 1; Proteinuria; Graft vs Host Disease; Kidney Failure, Chronic; Delayed Graft Function; Immune System Diseases; Kidney Transplantation
T-lymphocyte activation antigen CD80 inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY
ORAL
Adenocarcinoma; Carcinoma, Non-Small-Cell Lung; Esophageal Neoplasms; Hypertension; Renal Insufficiency; Schizophrenia; Stomach Neoplasms; Respiratory Tract Diseases; Severe Acute Respiratory Syndrome; Diabetes Mellitus; Diabetes Mellitus, Type 2
Dipeptidyl peptidase IV inhibitor
Protein
Approved
Unknown
Unknown
Heart Failure; Joint Diseases; Mitochondrial Diseases; Severe Acute Respiratory Syndrome; Angioedema; Angioedemas, Hereditary; Hypotension
Unknown
Protein
Approved
EYE
INJECTION
Carcinoma, Non-Small-Cell Lung; Corneal Neovascularization; Glioblastoma; Glioma; Histoplasmosis; Lymphoma; Lymphoma, Non-Hodgkin; Adenocarcinoma, Follicular; Astrocytoma; Brain Neoplasms; Breast Neoplasms; Carcinoid Tumor; Carcinoma, Renal Cell; Central Serous Chorioretinopathy; Colonic Neoplasms; Endometrial Neoplasms; Gliosarcoma; Graves Ophthalmopathy; Leukemia; Multiple Myeloma; Oligodendroglioma; Pseudoxanthoma Elasticum; Rectal Neoplasms; Retinal Diseases; Small Cell Lung Carcinoma; Thyroid Neoplasms; Urethral Neoplasms; Urinary Bladder Neoplasms; Uveal Melanoma; Vitreous Hemorrhage; Choroidal Neovascularization; Glaucoma; Glaucoma, Neovascular; Macular Degeneration; Melanoma; Retinopathy of Prematurity; Telangiectasis; Colorectal Neoplasms; Diabetes Complications; Diabetic Retinopathy; Macular Edema; Myopia, Degenerative; Neoplasms; Retinal Neovascularization; Retinal Vein Occlusion; Wet Macular Degeneration
Placenta growth factor inhibitor
Small molecule
Approved
Unknown
Unknown
Osteoarthritis, Knee
Unknown
Small molecule
Approved
Unknown
Unknown
Heart Arrest
Unknown
Small molecule
Approved
OTHER
INHALATION
Asthma; Lung Diseases; Bronchitis, Chronic; Emphysema; Pulmonary Disease, Chronic Obstructive
Beta-2 adrenergic receptor agonist
Small molecule
Approved
OTHER
TOPICAL
Lice Infestations
Nicotinic acetylcholine receptor agonist
Small molecule
Approved
Unknown
Unknown
Alcohol Drinking; Anxiety; Arthritis, Rheumatoid; Celiac Disease; Gingivitis; Otitis Media with Effusion; Acne Vulgaris; Amyotrophic Lateral Sclerosis; Burns; Chemical and Drug Induced Liver Injury; Hidradenitis Suppurativa; Ileus; Intervertebral Disc Degeneration; Melanoma; Severe Acute Respiratory Syndrome; Tinea Pedis; Cardiovascular Diseases; Dental Caries; Hemorrhoids; Infections; Pain; Periodontitis; Tension-Type Headache; Tooth Diseases
Unknown
Small molecule
Approved
Unknown
Unknown
Cardiovascular Diseases; Essential Hypertension; Hypertension
Unknown
Small molecule
Approved
OTHER
INTRAVENOUS
Arthritis, Rheumatoid; Cystitis, Interstitial; Genital Neoplasms, Female; Heart Failure; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Neoplasms; Central Nervous System Diseases
Diagnostic agent
Small molecule
Approved
Unknown
Unknown
Alzheimer Disease; Dementia; Lewy Body Disease; Movement Disorders; Multiple System Atrophy; Parkinson Disease; Parkinsonian Disorders; Radionuclide Imaging; Tomography, Emission-Computed, Single-Photon
Diagnostic agent
Antibody
Approved
DERMATOLOGY
INJECTION
Carcinoma, Pancreatic Ductal; Cholangiocarcinoma; Endometrial Neoplasms; Fallopian Tube Neoplasms; Glioma; HIV Infections; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Leukemia, Myeloid, Acute; Lymphoma; Lymphoma, Follicular; Lymphoma, Large B-Cell, Diffuse; Lymphoma, Non-Hodgkin; Multiple Myeloma; Myelodysplastic Syndromes; Neoplasm Metastasis; Nerve Sheath Neoplasms; Neuroblastoma; Peritoneal Neoplasms; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Retroperitoneal Neoplasms; Skin Neoplasms; Triple Negative Breast Neoplasms; Adenocarcinoma; Adenocarcinoma of Lung; Basal Cell Nevus Syndrome; Biliary Tract Neoplasms; Breast Neoplasms; Carcinoid Tumor; Carcinoma; Carcinoma, Basal Cell; Carcinoma, Merkel Cell; Carcinoma, Neuroendocrine; Carcinoma, Small Cell; Colonic Neoplasms; Esophageal Neoplasms; Gastrointestinal Stromal Tumors; Gliosarcoma; Histiocytoma, Malignant Fibrous; Hodgkin Disease; Inflammatory Breast Neoplasms; Leiomyosarcoma; Liposarcoma; Meningioma; Nasopharyngeal Carcinoma; Neuroendocrine Tumors; Ovarian Neoplasms; Pancreatic Neoplasms; Pituitary Neoplasms; Prostatic Neoplasms; Rectal Neoplasms; Retroviridae Infections; Salivary Gland Neoplasms; Sarcoma, Kaposi; Sarcoma, Synovial; Urinary Bladder Neoplasms; Uterine Cervical Neoplasms; Uveal Melanoma; Carcinoma, Hepatocellular; Carcinoma, Squamous Cell; Glioblastoma; Head and Neck Neoplasms; Kidney Neoplasms; Lung Neoplasms; Mesothelioma; Prostatic Neoplasms, Castration-Resistant; Sarcoma; Small Cell Lung Carcinoma; Stomach Neoplasms; Urogenital Neoplasms; Carcinoma, Non-Small-Cell Lung; Carcinoma, Renal Cell; Colorectal Neoplasms; Melanoma; Mesothelioma, Malignant; Neoplasms
Cytotoxic T-lymphocyte protein 4 inhibitor
Small molecule
Approved
DERMATOLOGY
ORAL
Lymphoma; Paraganglioma; Skin Neoplasms; Carcinoma, Non-Small-Cell Lung; Colorectal Neoplasms; Craniopharyngioma; Hematologic Neoplasms; Histiocytosis; Histiocytosis, Langerhans-Cell; Leukemia, Hairy Cell; Leukemia, Myeloid, Acute; Multiple Myeloma; Pancreatic Neoplasms; Thyroid Neoplasms; Melanoma; Neoplasms
Serine/threonine-protein kinase B-raf inhibitor
Unknown
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
Unknown
Unknown
Lung Diseases; Asthma; Heart Failure; Pulmonary Disease, Chronic Obstructive; Lung Diseases, Obstructive
Unknown
Small molecule
Approved
DERMATOLOGY; NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Kidney Diseases; Alcoholism; Diabetic Neuropathies; Migraine Disorders; Neuralgia, Postherpetic; Restless Legs Syndrome
Voltage-gated calcium channel modulator
Small molecule
Approved
RESPIRATORY
ORAL
Multiple Sclerosis; Acute Lung Injury; Alveolitis, Extrinsic Allergic; Bronchiolitis Obliterans; Burns; Carcinoma, Squamous Cell; Cardiomyopathy, Hypertrophic; Glomerulosclerosis, Focal Segmental; Heart Failure; Leiomyoma; Lung Diseases, Interstitial; Lung Neoplasms; Nephrotic Syndrome; Neurofibromatosis 1; Pancreatitis; Proteinuria; Pulmonary Fibrosis; Radiation Pneumonitis; Renal Insufficiency; Renal Insufficiency, Chronic; Scleroderma, Systemic; Diabetic Foot; Keloid; Pneumoconiosis; Pneumonia; Respiratory Distress Syndrome; Severe Acute Respiratory Syndrome; Idiopathic Pulmonary Fibrosis; Immune System Diseases; Lung Diseases; Respiratory Tract Diseases
Unknown
Small molecule
Approved
IMMUNE SYSTEM
ORAL
Thrombocytopenia; Hepatitis C; Hepatitis C, Chronic; Virus Diseases
Hepatitis C virus serine protease, NS3/NS4A inhibitor
Small molecule
Approved
Unknown
Unknown
Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Neoplasms
Androgen Receptor antagonist
Small molecule
Approved
Unknown
Unknown
Carcinoma, Pancreatic Ductal; Dermatitis; Glioblastoma; Leukemia, Biphenotypic, Acute; Lung Neoplasms; Lymphoma, Non-Hodgkin; Malignant Atrophic Papulosis; Neuromyelitis Optica; Paraganglioma; Pneumonia; Uveal Melanoma; Alopecia Areata; Anemia; Arthritis, Rheumatoid; beta-Thalassemia; Breast Neoplasms; Bronchiolitis Obliterans; Bronchiolitis Obliterans Syndrome; Cachexia; Carcinoma, Non-Small-Cell Lung; Carcinoma, Squamous Cell; Colorectal Neoplasms; Dermatitis, Seborrheic; Hematologic Neoplasms; Hidradenitis Suppurativa; Histiocytosis; HIV Infections; Hodgkin Disease; Hypereosinophilic Syndrome; Inflammatory Breast Neoplasms; Leukemia; Leukemia, Large Granular Lymphocytic; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid, Acute; Lichen Planus; Lichen Sclerosus et Atrophicus; Lupus Erythematosus, Discoid; Lymphoma; Multiple Myeloma; Necrobiosis Lipoidica; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Primary Immunodeficiency Diseases; Prostatic Neoplasms, Castration-Resistant; Psoriasis; Dermatitis, Atopic; Graft vs Host Disease; Lymphohistiocytosis, Hemophagocytic; Macrophage Activation Syndrome; Myeloproliferative Disorders; Pancreatic Neoplasms; Polycythemia Vera; Primary Myelofibrosis; Prurigo; Severe Acute Respiratory Syndrome; Thrombocythemia, Essential; Vitiligo; Eczema; Neoplasms
Unknown
Protein
Approved
GASTROINTESTINAL
ORAL
Liver Diseases; Thrombocytopenia; Hepatitis C; HIV Infections; Infections; Hepatitis C, Chronic; Virus Diseases
Hepatitis C virus serine protease, NS3/NS4A inhibitor
Small molecule
Approved
OTHER; UROLOGY AND KIDNEY
ORAL
Kidney Diseases; Erectile Dysfunction
Phosphodiesterase 5A inhibitor
Small molecule
Approved
OTHER
ORAL
Hepatitis C; Insulin Resistance; Acquired Immunodeficiency Syndrome; HIV Infections; Virus Diseases
Human immunodeficiency virus type 1 reverse transcriptase inhibitor
Small molecule
Approved
Unknown
Unknown
Marijuana Abuse; Memory Disorders; Anxiety Disorders; Depressive Disorder
Unknown
Small molecule
Approved
Unknown
Unknown
Brain Diseases; Depressive Disorder, Major; Lymphoma; Neoplasms; Nervous System Diseases; Obesity; Peripheral Nervous System Diseases; Schizophrenia; Cognitive Dysfunction; Dementia; Dermatitis; Dermatitis, Seborrheic; Diabetes Mellitus, Type 2; Fragile X Syndrome; Non-alcoholic Fatty Liver Disease; Respiratory Distress Syndrome; Rosacea; Asthma; Bronchiectasis; Dermatitis, Atopic; Diabetic Nephropathies; Bronchitis, Chronic; Lung Diseases, Obstructive; Psoriasis; Pulmonary Disease, Chronic Obstructive
Phosphodiesterase 4 inhibitor
Small molecule
Approved
DIABETES DRUGS & ENDOCRINOLOGY; OTHER
ORAL
Polycystic Ovary Syndrome; Renal Insufficiency; Breast Neoplasms; Diabetes Mellitus, Type 1; Obesity; Renal Insufficiency, Chronic; Diabetic Nephropathies; Heart Failure; Diabetes Mellitus; Diabetes Mellitus, Type 2
Sodium/glucose cotransporter 2 inhibitor
Small molecule
Approved
GASTROINTESTINAL
ORAL
Clostridium Infections; Diarrhea; Infections
DNA-directed RNA polymerase inhibitor
Small molecule
Approved
NEUROLOGY DRUGS & NERVOUS SYSTEM; OTHER
ORAL
Amyotrophic Lateral Sclerosis; Depressive Disorder; Depressive Disorder, Major; Neuralgia, Postherpetic; Epilepsy; Seizures
KCNQ (Kv7) potassium channel opener
Small molecule
Approved
Unknown
Unknown
Unknown
Unknown
Small molecule
Approved
CARDIOVASCULAR; HEMATOLOGY; OTHER
ORAL
Blood Coagulation Disorders; Obesity, Morbid; Renal Insufficiency, Chronic; Anemia, Sickle Cell; Aortic Valve Disease; Heart Diseases; Hemorrhage; Ischemia; Multiple Myeloma; Thromboembolism; Angina, Unstable; Aortic Valve Stenosis; Diabetes Mellitus, Type 2; Hematoma; Hip Fractures; Ischemic Stroke; Liver Cirrhosis; Myocardial Infarction; Neoplasms; Polyendocrinopathies, Autoimmune; Renal Insufficiency; Rheumatic Heart Disease; Severe Acute Respiratory Syndrome; Thrombocytopenia; Acute Coronary Syndrome; Arthroplasty, Replacement; Atrial Fibrillation; Coronary Artery Disease; Peripheral Arterial Disease; Pulmonary Embolism; Stroke; Thrombosis; Venous Thromboembolism; Venous Thrombosis
Coagulation factor X inhibitor
Small molecule
Approved
CARDIOVASCULAR; OTHER
ORAL
Hypertension; Stroke
Type-1 angiotensin II receptor antagonist
Antibody
Approved
CANCER; OTHER
INJECTION
Hematologic Neoplasms; HIV Infections; Leukemia; Leukemia, Myeloid, Acute; Enteropathy-Associated T-Cell Lymphoma; Graft vs Host Disease; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Mast-Cell; Lupus Erythematosus, Systemic; Lymphoma, Follicular; Lymphoma, T-Cell, Peripheral; Mastocytosis, Systemic; Mesothelioma, Malignant; Neoplasms, Germ Cell and Embryonal; Scleroderma, Diffuse; Sezary Syndrome; Lymphoma; Lymphoma, Large B-Cell, Diffuse; Lymphoma, T-Cell, Cutaneous; Mycosis Fungoides; Hodgkin Disease; Lymphoma, Large-Cell, Anaplastic; Lymphoma, Non-Hodgkin; Neoplasms
Tubulin inhibitor
Enzyme
Approved
Unknown
Unknown
Leukemia, Lymphoid; Neoplasms; Leukemia, Biphenotypic, Acute; Myelodysplastic Syndromes; Leukemia; Leukemia, Myeloid, Acute; Precursor Cell Lymphoblastic Leukemia-Lymphoma
Asparagine hydrolytic enzyme
Antibody
Approved
Unknown
Unknown
Graft vs Host Disease; Lymphopenia; Neuromyelitis Optica; Arthritis, Rheumatoid; Emphysema; Glomerulonephritis, Membranous; Kidney Diseases; Leukemia, Lymphocytic, Chronic, B-Cell; Multiple Sclerosis; Myositis; Nephrotic Syndrome; Polyendocrinopathies, Autoimmune; Scleroderma, Systemic; Sjogren's Syndrome; Purpura, Thrombocytopenic, Idiopathic; Vasculitis; Lupus Erythematosus, Systemic; Lupus Nephritis
Tumor necrosis factor ligand superfamily member 13B inhibitor